4ivc B 2.35 BS01 1J6 B 1 L881 G882 E883 V889 A906 M956 F958 L959 E966 L1010 D1021 L17 G18 E19 V25 A42 M84 F86 L87 E94 L138 D149 D1003 A1005 R1007 N1008 D1021 D1040 D131 A133 R135 N136 D149 D168 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.1nM EC50=28nM, IC50=<0.200nM, Ki=0.100000nM P23458 23659214 1201 VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTNGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK