4ith B 2.25 BS01 RCM B 1 M67 L70 V75 V76 L78 M92 A155 D156 S161 F162 M55 L58 V63 V64 L66 M80 A143 D144 S149 F150 D138 K140 E142 N143 D156 T189 D126 K128 E130 N131 D144 T165 2.7.11.1 0004672,0005524,0006468 ic50=0.3169uM IC50=200nM, EC50=18nM Q13546 23473668 307 LNVIKMKSSDFLESAELKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNEGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE