4h82 B 1.9 BS01 L29 A 1 L187 L188 A189 H190 L222 H226 Q227 H230 H236 L243 Y245 P246 M247 L78 L79 A80 H81 L113 H117 Q118 H121 H127 L134 Y136 P137 M138 H226 Q227 H230 H236 H117 Q118 H121 H127 3.4.24.35 0004222,0006508,0008237,0008270,0031012 IC50=5.5nM P14780 23567804 306 FEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h82 B 1.9 BS02 ZN B 1 H226 H230 H236 H117 H121 H127 H226 Q227 H230 H236 H117 Q118 H121 H127 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 300 FEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h82 B 1.9 BS03 ZN B 2 H175 D177 H190 H203 H66 D68 H81 H94 H226 Q227 H230 H236 H117 Q118 H121 H127 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 301 FEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h82 B 1.9 BS04 CA B 1 D165 G197 Q199 D201 D56 G88 Q90 D92 H226 Q227 H230 H236 H117 Q118 H121 H127 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 302 FEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h82 B 1.9 BS05 CA B 2 D182 G183 K184 D185 L187 D205 E208 D73 G74 K75 D76 L78 D96 E99 H226 Q227 H230 H236 H117 Q118 H121 H127 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 303 FEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG 4h82 B 1.9 BS06 CA B 3 D131 D206 E208 D22 D97 E99 H226 Q227 H230 H236 H117 Q118 H121 H127 3.4.24.35 0004222,0006508,0008237,0008270,0031012 P14780 23567804 304 FEGDLKWHHHNITYWIQNYSEDLPRAVIDDAFARAFALWSAVTPLTFTRVYSRDADIVIQFGVAEHGDGYPFDGKDGLLAHAFPPGPGIQGDAHFDDDELWSLGKGQGYSLFLVAAHQFGHALGLDHSSVPEALMYPMYRFTEGPPLHKDDVNGIRHLYG