4dbn B 3.15 BS01 0JA B 1 A480 K482 E500 V503 L504 L513 I526 T528 W530 C531 F582 G592 D593 F594 A34 K36 E54 V57 L58 L67 I80 T82 W84 C85 F136 G146 D147 F148 D575 K577 N579 N580 D593 W603 S615 D129 K131 N133 N134 D147 W157 S159 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=8.15, IC50=7.0nM P15056 22376051 901 DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS