4bbe B 1.9 BS01 3O4 B 1 L855 G856 V863 Y931 L932 G935 L983 L15 G16 V23 Y91 L92 G95 L143 N976 A978 R980 N981 D994 S1016 N136 A138 R140 N141 D154 S176 2.7.10.2 0004672,0005524,0006468 ic50=3.6nM IC50=974.7nM O60674 23127890 2229 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRNLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRD