3ri1 B 2.1 BS01 3RH B 1 V495 A515 K517 M538 V564 A567 L633 V28 A45 K47 M68 V94 A97 L150 D626 A628 R630 N631 D644 D143 A145 R147 N148 D161 2.7.10.1 0004672,0004713,0005524,0006468 Kd=5uM IC50=1230nM P21802 21454610 1 LPEDPKWEFPRDKLTLGKPLGEGCFGQVVMAEAVGIDPKEAVTVAVKMLKDDATEKDLSDLVSEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLRARRPPEQMTFKDLVSCTYQLARGMEYLASQKCIHRDLAARNVLVTENNVMKIADFGLARDINNIDYYKKTTNGRLPVKWMAPEALFDRVYTHQSDVWSFGVLMWEIFTLGGSPYPGIPVEELFKLLKEGHRMDKPANCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRILTLTTN