3qs1 B 3.1 BS01 006 B 1 D32 G34 N74 Y75 V76 S77 L128 D215 G217 T218 S219 I300 D33 G35 N75 Y76 V77 S78 L130 D213 G215 T216 S217 I299 D32 S35 N37 W39 Y75 D215 T218 D33 S36 N38 W40 Y76 D213 T216 3.4.23.38 0004190,0006508 -logKd/Ki=7.96, Ki=11.0nM IC50=280nM P39898 21521654 330 AGDSVTLNDVANVMYYGEAQIGDNKQKFAFIFDTGSANLWVPSAQCNTIGCKTKNLYDSNKSKTYEKDGTKVEMNYVSGTVSGFFSKDIVTIANLSFPYKFIEVTDTNGFEPAYTLGQFDGIVGLGWKDLSIGSVDPVVVELKNQNKIEQAVFTFYLPFDDKHKGYLTIGGIEDRFYEGQLTYEKLNHDLYWQVDLDLHFGNLTVEKATAIVDSGTSSITAPTEFLNKFFEGLDVVKIPFLPLYITTCNNPKLPTLEFRSATNVYTLEPEYYLQQIFDFGISLCMVSIIPVDLNKNTFILGDPFMRKYFTVFDYDNHTVGFALAKKK