3idp B 2.7 BS01 L1E B 1 V471 A481 K483 E501 L505 L514 T529 W531 C532 F583 G593 D594 F595 V23 A33 K35 E53 L57 L66 T81 W83 C84 F135 G145 D146 F147 D576 K578 N580 N581 D594 S616 D128 K130 N132 N133 D146 S152 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=8.80, IC50=1.6nM Ki=1nM, IC50=2nM P15056 19764794 1 DWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKIGDFGLSGSILWMAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLARS