3fq7 A 2.15 BS02 PXG B 1 G1304 T1305 G298 T299 V1027 Y1150 D1245 M1248 K1273 A1407 V21 Y144 D239 M242 K267 A401 5.4.3.8 0005737,0006782,0008483,0015995,0016853,0030170,0033014,0042286 -logKd/Ki=2.52, IC50=3mM P24630 19786580 2434 FKTIKSDEIFAAAQKLMPGGVSSPVRAFKSVGGQPIVFDRVKDAYAWDVDGNRYIDYVGTWGPAICGHAHPEVIEALKVAMEKGTSFGAPCALENVLAEMVNDAVPSIEMVRFVNSGTEACMAVLRIMRAYTGRDKIIKFEGCYHGHADMFLVKAGSGVATLGLPSSPGVPKKTTANTLTTPYNDLEAVKALFAENPGEIAGVILEPIVGNSGFIVPDAGFLEGLREITLEHDALLVFDEVMTGFRIAYGGVQEKFGVTPDLTTLGKIIGGGLPVGAYGGKREIMQLVAPAGPMYQAGTLSGNPLAMTAGIKTLELLRQPGTYEYLDQITKRLSDGLLAIAQETGHAACGGQVSGMFGFFFTEGPVHNYEDAKKSDLQKFSRFHRGMLEQGIYLAPSQFEAGFTSLAHTEEDIDATLAAARTVMSAL 3fq7 B 2.15 BS01 PXG A 1 A2303 G2304 T2305 A297 G298 T299 V2027 Y2150 E2212 D2245 M2248 K2273 A2407 V21 Y144 E206 D239 M242 K267 A401 5.4.3.8 0005737,0006782,0008483,0015995,0016853,0030170,0033014,0042286 -logKd/Ki=2.52, IC50=3mM P24630 19786580 1434 FKTIKSDEIFAAAQKLMPGGVSSPVRAFKSVGGQPIVFDRVKDAYAWDVDGNRYIDYVGTWGPAICGHAHPEVIEALKVAMEKGTSFGAPCALENVLAEMVNDAVPSIEMVRFVNSGTEACMAVLRIMRAYTGRDKIIKFEGCYHGHADMFLVKAGSGVATLGLPSSPGVPKKTTANTLTTPYNDLEAVKALFAENPGEIAGVILEPIVGNSGFIVPDAGFLEGLREITLEHDALLVFDEVMTGFRIAYGGVQEKFGVTPDLTTLGKIIGGGLPVGAYGGKREIMQLVAPAGPMYQAGTLSGNPLAMTAGIKTLELLRQPGTYEYLDQITKRLSDGLLAIAQETGHAACGGQVSGMFGFFFTEGPVHNYEDAKKSDLQKFSRFHRGMLEQGIYLAPSQFEAGFTSLAHTEEDIDATLAAARTVMSAL 3fq7 B 2.15 BS02 PXG B 1 S2029 V2031 W2067 S2122 G2123 T2124 Y2150 H2151 E2212 N2217 D2245 V2247 M2248 K2273 E2406 S23 V25 W61 S116 G117 T118 Y144 H145 E206 N211 D239 V241 M242 K267 E400 V2027 Y2150 E2212 D2245 M2248 K2273 A2407 V21 Y144 E206 D239 M242 K267 A401 5.4.3.8 0005737,0006782,0008483,0015995,0016853,0030170,0033014,0042286 -logKd/Ki=2.52, IC50=3mM P24630 19786580 2434 FKTIKSDEIFAAAQKLMPGGVSSPVRAFKSVGGQPIVFDRVKDAYAWDVDGNRYIDYVGTWGPAICGHAHPEVIEALKVAMEKGTSFGAPCALENVLAEMVNDAVPSIEMVRFVNSGTEACMAVLRIMRAYTGRDKIIKFEGCYHGHADMFLVKAGSGVATLGLPSSPGVPKKTTANTLTTPYNDLEAVKALFAENPGEIAGVILEPIVGNSGFIVPDAGFLEGLREITLEHDALLVFDEVMTGFRIAYGGVQEKFGVTPDLTTLGKIIGGGLPVGAYGGKREIMQLVAPAGPMYQAGTLSGNPLAMTAGIKTLELLRQPGTYEYLDQITKRLSDGLLAIAQETGHAACGGQVSGMFGFFFTEGPVHNYEDAKKSDLQKFSRFHRGMLEQGIYLAPSQFEAGFTSLAHTEEDIDATLAAARTVMSAL