2wtv B 2.4 BS01 ZZL B 1 L139 K141 V147 K162 Y212 A213 G216 L263 A273 D274 V279 L14 K16 V22 K37 Y87 A88 G91 L138 A148 D149 V154 D256 K258 E260 N261 D274 T292 D131 K133 E135 N136 D149 T167 2.7.11.1 0000212,0000226,0000278,0004672,0005524,0006468,0007052,0007098,0007100,0051321 Ki=1.8nM IC50=34nM, Kd=6.5nM O14965 20067443 1390 RQWALEDFEIGRPLGKGKFGNVYLAREKQSKFILALKVLFKAQLEKAGVEHQLRREVEIQSHLRHPNILRLYGYFHDATRVYLILEYAPRGEVYKELQKLSKFDEQRTATYITELANALSYCHSKRVIHRDIKPENLLLGSAGELKIADFGWSVHAPSSRRTTLCGTLDYLPPEMIEGRMHDEKVDLWSLGVLCYEFLVGKPPFEANTYQETYKRISRVEFTFPDFVTEGARDLISRLLKHNPSQRPMLREVLEHPWITANSSK