2q5p B 2.3 BS01 241 B 1 F226 G284 C285 R288 S289 A292 I326 Y327 M329 L330 L333 L340 I341 S342 F363 F20 G62 C63 R66 S67 A70 I104 Y105 M107 L108 L111 L118 I119 S120 F141 ? 0003677,0004879,0005634,0006355 IC50=1nM, EC50=2.0nM P37231 17937915 7001 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKSPFVIYDMNSLMMGEFKHITVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVILHPLLQEIYKD