2p4i B 2.5 BS01 MR9 B 1 K855 E872 L876 I886 I902 Y904 A905 F960 H962 L971 I980 A981 D982 F983 K15 E29 L33 I43 I55 Y57 A58 F113 H115 L124 I133 A134 D135 F136 D964 A966 R968 N969 D982 R999 D117 A119 R121 N122 D135 R140 2.7.10.1 0004672,0004713,0005524,0006468 ic50=10nM IC50=10nM Q02763 17253678 302 GQVLKARIRMDAAIKRMKEKDDHRDFAGELEVLCKLGHHPNIINLLGACEHYLAIEYAPHGNLLDFLRKSRVLETDPAFAIANSTASTLSSQQLLHFAADVARGMDYLSQKQFIHRDLAARNILVGENYVAKIADFGLGRLPVRWMAIESLNYSVYTTNSDVWSYGVLLWEIVSLGGTPYCGMTCAELYEKLPQGYRLEKPLNCDDEVYDLMRQCWREKPYERPSFAQILVSLNRMLEERKTYVNTTLYEKFTYAGID