2g0h B 2.3 BS01 SP3 B 1 I281 F282 C285 Q286 R288 S289 Y327 F363 M364 H449 I75 F76 C79 Q80 R82 S83 Y121 F157 M158 H243 ? 0003677,0004879,0005634,0006355 ic50=22.7nM IC50=23nM, EC50=0.78nM P37231 16640330 201 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLY