2e2b B 2.2 BS01 406 B 1 L248 Y253 V256 A269 K271 E286 V289 M290 L298 I313 T315 F317 M318 I360 H361 R362 A380 D381 F382 L24 Y29 V32 A45 K47 E57 V60 M61 L69 I84 T86 F88 M89 I131 H132 R133 A151 D152 F153 D363 A365 R367 N368 D381 P402 D134 A136 R138 N139 D152 P167 2.7.10.2 0004672,0004713,0005524,0006468 ic50=11nM IC50=4.0nM P00519 17376680 1002 MDPSSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMF