1uum B 2.3 BS01 FMN B 1 A95 A96 G97 K100 S120 N145 Y147 N181 N212 K255 N284 T285 S305 G306 V333 G334 G335 L355 Y356 T357 A58 A59 G60 K63 S83 N108 Y110 N144 N175 K209 N238 T239 S259 G260 V287 G288 G289 L309 Y310 T311 G119 N145 F149 S215 K255 N284 G82 N108 F112 S178 K209 N238 1.3.5.2 0004151,0004152,0005737,0005739,0005743,0006207,0006221,0006225,0007565,0007595,0009220,0009410,0010181,0014070,0016020,0016491,0016627,0031000,0042594,0043025,0043065,0044205,0048038,0048039,0090140,0106430,1903576 Q63707 15044733 398 YAEYLMPGLQRLLDPESAHRLAVRVTSLGLLPRATFQDSDMLEVKVLGHKFRNPVGIAAGFDKNGEAVDGLYKLGFGFVEVGSVTPQPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAQLTADGLPLGINLGKNKTSEDAAADYAEGVRTLGPLADYLVVNVSSQGKTELRHLLSKVLQERDALKGTRKPAVLVKIAPDLTAQDKEDIASVARELGIDGLIVTNTTVSRPVGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRIPIIGVGGVSSGQDALEKIQAGASLVQLYTALIFLGPPVVVRVKRELEALLKERGFTTVTDAIGADHRR 1uum B 2.3 BS02 AFI B 1 E40 M43 P44 Q47 P52 A55 H56 V134 R136 Y356 I360 P364 E3 M6 P7 Q10 P15 A18 H19 V97 R99 Y310 I314 P318 G119 N145 F149 S215 K255 N284 G82 N108 F112 S178 K209 N238 1.3.5.2 0004151,0004152,0005737,0005739,0005743,0006207,0006221,0006225,0007565,0007595,0009220,0009410,0010181,0014070,0016020,0016491,0016627,0031000,0042594,0043025,0043065,0044205,0048038,0048039,0090140,0106430,1903576 ic50=698nM Q63707 15044733 400 YAEYLMPGLQRLLDPESAHRLAVRVTSLGLLPRATFQDSDMLEVKVLGHKFRNPVGIAAGFDKNGEAVDGLYKLGFGFVEVGSVTPQPQEGNPRPRVFRLPEDQAVINRYGFNSHGLSVVEHRLRARQQKQAQLTADGLPLGINLGKNKTSEDAAADYAEGVRTLGPLADYLVVNVSSQGKTELRHLLSKVLQERDALKGTRKPAVLVKIAPDLTAQDKEDIASVARELGIDGLIVTNTTVSRPVGLQGALRSETGGLSGKPLRDLSTQTIREMYALTQGRIPIIGVGGVSSGQDALEKIQAGASLVQLYTALIFLGPPVVVRVKRELEALLKERGFTTVTDAIGADHRR