1mx1 B 2.4 BS01 SIA A 1 K2262 T2278 K241 T257 G2142 G2143 S2221 A2222 E2354 H2468 G121 G122 S200 A201 E333 H446 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 P23141 12725862 182 SPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK 1mx1 B 2.4 BS02 SIA B 1 L2051 G2052 K2078 N2079 A2080 T2081 S2082 P2084 Y2118 L30 G31 K57 N58 A59 T60 S61 P63 Y97 G2142 G2143 S2221 A2222 E2354 H2468 G121 G122 S200 A201 E333 H446 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 P23141 12725862 282 SPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK 1mx1 B 2.4 BS03 THA B 1 S2221 L2304 L2363 S200 L283 L341 G2142 G2143 S2221 A2222 E2354 H2468 G121 G122 S200 A201 E333 H446 3.1.1.1,3.1.1.13,3.1.1.56 0004771,0005737,0005783,0005788,0005811,0005829,0006629,0006695,0008203,0009636,0010875,0010887,0016042,0030855,0042632,0043691,0047374,0051791,0052689,0070857,0071397,0071404,0090122,0090205,0106435,0120188 IC50=>100000nM, Ki=>100000nM P23141 12725862 2 SPPVVDTVHGKVLGKFVSLEGFAQPVAIFLGIPFAKPPLGPLRFTPPQPAEPWSFVKNATSYPPMCTQDPKAGQLLSELFTNRKENIPLKLSEDCLYLNIYTPADLTKKNRLPVMVWIHGGGLMVGAASTYDGLALAAHENVVVVTIQYRLGIWGFFSTGDEHSRGNWGHLDQVAALRWVQDNIASFGGNPGSVTIFGESAGGESVSVLVLSPLAKNLFHRAISESGVALTSVLVKKGDVKPLAEQIAITAGCKTTTSAVMVHCLRQKTEEELLETTLKMKFLSLDLQGDPRESQPLLGTVIDGMLLLKTPEELQAERNFHTVPYMVGINKQEFGWLIPMLMSYPLSEGQLDQKTAMSLLWKSYPLVCIAKELIPEATEKYLGGTDDTVKKKDLFLDLIADVMFGVPSVIVARNHRDAGAPTYMYEFQYRPSFSSDMKPKTVIGDHGDELFSVFGAPFLKEGASEEEIRLSKMVMKFWANFARNGNPNGEGLPHWPEYNQKEGYLQIGANTQAAQKLKDKEVAFWTNLFAK