1iyk B 2.3 BS01 MYA B 1 Y107 V108 I174 L177 I179 R184 N185 R187 A189 P190 I193 T197 A208 Y210 I215 L216 Y48 V49 I115 L118 I120 R125 N126 R128 A130 P131 I134 T138 A149 Y151 I156 L157 N175 F176 L177 T211 L451 N116 F117 L118 T152 L392 2.3.1.97 0004379,0006499 P30418 12401496 1501 EGPIDKLKTPEDVPNDPLPLISDFEWSTLDIDDNLQLDELYKLLYDNYVEDIDATFRFKYSHEFFQWALKPPGWRKDWHVGVRVKSTGKLVAFIAATPVTFKLNKSNKVIDSVEINFLCIHKKLRNKRLAPVLIKEITRRVNKQNIWQALYTGGSILPTPLTTCRYQHRPINWSKLHDVGFSHLPPNQTKSSMVASYTLPNNPKLKGLRPMTGKDVSTVLSLLYKYQERFDIVQLFTEEEFKHWMLGHDENSDSNVVKSYVVEDENGIITDYFSYYLLPFTVLDNAQHDELGIAYLFYYASDSFEKPNYKKRLNELITDALITSKKFGVDVFNCLTCQDNTYFLKDCKFGSGDGFLNYYLFNYRTFPMDGGIDKKTKEVVEDQTSGIGVVLL 1iyk B 2.3 BS02 MIM B 1 V108 D110 F115 F117 T211 Y225 H227 P229 F240 F339 G409 G411 D412 G413 L451 V49 D51 F56 F58 T152 Y166 H168 P170 F181 F280 G350 G352 D353 G354 L392 N175 F176 L177 T211 L451 N116 F117 L118 T152 L392 2.3.1.97 0004379,0006499 Ki=0.25uM Ki=31nM P30418 12401496 1502 EGPIDKLKTPEDVPNDPLPLISDFEWSTLDIDDNLQLDELYKLLYDNYVEDIDATFRFKYSHEFFQWALKPPGWRKDWHVGVRVKSTGKLVAFIAATPVTFKLNKSNKVIDSVEINFLCIHKKLRNKRLAPVLIKEITRRVNKQNIWQALYTGGSILPTPLTTCRYQHRPINWSKLHDVGFSHLPPNQTKSSMVASYTLPNNPKLKGLRPMTGKDVSTVLSLLYKYQERFDIVQLFTEEEFKHWMLGHDENSDSNVVKSYVVEDENGIITDYFSYYLLPFTVLDNAQHDELGIAYLFYYASDSFEKPNYKKRLNELITDALITSKKFGVDVFNCLTCQDNTYFLKDCKFGSGDGFLNYYLFNYRTFPMDGGIDKKTKEVVEDQTSGIGVVLL