1g05 B 2.45 BS01 ZN B 1 H701 H705 H711 H119 H123 H129 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 P08254 11327577 801 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHFRLSQDDINGIQSLYGPPPDSPET 1g05 B 2.45 BS02 ZN B 2 H651 D653 H666 H679 H69 D71 H84 H97 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 P08254 11327577 802 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHFRLSQDDINGIQSLYGPPPDSPET 1g05 B 2.45 BS03 CA B 1 D658 G659 G661 V663 D681 E684 D76 G77 G79 V81 D99 E102 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 P08254 11327577 803 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHFRLSQDDINGIQSLYGPPPDSPET 1g05 B 2.45 BS04 CA B 2 D607 D682 E684 D25 D100 E102 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 P08254 11327577 804 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHFRLSQDDINGIQSLYGPPPDSPET 1g05 B 2.45 BS05 CA B 3 D641 G673 N675 D677 D59 G91 N93 D95 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 P08254 11327577 805 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHFRLSQDDINGIQSLYGPPPDSPET 1g05 B 2.45 BS06 BBH B 1 N662 L664 A665 H701 E702 H705 H711 N80 L82 A83 H119 E120 H123 H129 H701 E702 H705 H711 H119 E120 H123 H129 3.4.24.17 0004222,0006508,0008237,0008270,0031012 ic50=3.1nM -logKd/Ki=8.51, IC50=3.1nM IC50=3.1nM P08254 11327577 901 FRTFPGIPKWRKTHLTYRIVNYTPDLPKDAVDSAVEKALKVWEEVTPLTFSRLYEGEADIMISFAVREHGDFYPFDGPGNVLAHAYAPGPGINGDAHFDDDEQWTKDTTGTNLFLVAAHEIGHSLGLFHSANTEALMYPLYHFRLSQDDINGIQSLYGPPPDSPET