1fgi B 2.5 BS01 SU1 B 1 G485 F489 A512 Y563 A564 G567 L630 G25 F29 A48 Y99 A100 G103 L150 D623 A625 R627 N628 D641 D143 A145 R147 N148 D161 2.7.10.1 0004672,0004713,0005007,0005524,0006468 IC50=30nM P11362 9139660 1000 SEYELPEDPRWELPRDRLVLGKPLGEGAFGQVVLAEAIGLPNRVTKVAVKMLKSDATEKDLSDLISEMEMMKMIGKHKNIINLLGACTQDGPLYVIVEYASKGNLREYLQARRQLSSKDLVSCAYQVARGMEYLASKKCIHRDLAARNVLVTEDNVMKIADFGLADYYKKGRLPVKWMAPEALFDRIYTHQSDVWSFGVLLWEIFTLGGSPYPGVPVEELFKLLKEGHRMDKPSNCTNELYMMMRDCWHAVPSQRPTFKQLVEDLDRIVALT