6s9x A 2.6 BS01 L1W A 1 Q79 W80 I84 L210 L264 V270 Y272 R273 D292 C296 C310 Q73 W74 I78 L156 L210 V216 Y218 R219 D238 C242 C249 D274 K276 N279 D292 T312 D220 K222 N225 D238 T251 2.7.11.1 0001649,0001893,0001934,0001938,0002042,0003376,0004672,0004674,0004712,0005515,0005516,0005524,0005547,0005634,0005654,0005737,0005739,0005758,0005819,0005829,0005886,0005911,0005938,0005977,0005978,0005979,0006006,0006338,0006417,0006468,0006469,0006606,0006809,0006915,0006924,0006954,0006979,0007165,0007173,0007186,0007281,0007399,0008283,0008286,0008637,0009408,0009725,0010467,0010507,0010595,0010628,0010629,0010748,0010761,0010763,0010765,0010907,0010951,0010975,0015630,0016020,0016242,0016301,0016310,0016567,0018105,0018107,0019049,0019221,0019899,0019901,0022605,0030027,0030154,0030163,0030235,0030291,0030307,0030334,0030335,0031295,0031397,0031641,0031663,0031929,0031982,0031999,0032079,0032091,0032094,0032287,0032436,0032869,0032880,0032991,0033138,0034405,0035556,0035655,0035924,0036064,0036294,0042593,0042802,0042803,0042981,0043066,0043154,0043161,0043276,0043325,0043488,0043491,0043536,0044024,0045429,0045600,0045725,0045737,0045746,0045861,0045944,0046326,0046622,0046777,0046889,0048009,0048266,0048661,0051000,0051091,0051146,0051247,0060079,0060416,0060644,0060709,0060716,0070141,0070848,0071356,0071363,0071364,0071380,0071889,0071901,0072655,0072656,0072752,0090201,0097011,0097194,0098794,0098978,0099104,0099175,0106310,0110002,0140052,0150033,0160049,1900087,1900182,1901653,1901796,1902018,1902176,1903038,1903078,1903318,1904263,1905552,1990090,1990418,2000010,2000074,2000402,2001240,2001243 -logKd/Ki=6.42, IC50=381nM P31749 31584233 501 DVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDEAPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGLKRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPKQRLGGGSEDAKEIMQHRFFAGIVWQHVYEKKLSPPFKPQVTSETDTRYFDEEFT