6rtn A 2.17 BS01 KJK A 1 S67 K70 S115 V117 T206 G207 F208 R250 S48 K51 S96 V98 T187 G188 F189 R231 S67 K70 S115 F120 W154 F208 S48 K51 S96 F101 W135 F189 3.5.2.6 0008658,0008800,0017001 -logKd/Ki=6.63, IC50=0.234uM P14489 31454231 506 GSITENTSWNKEFSAEAVNGVFVLCKSSSKSCATNDLARASKEYLPASTFKIPNAIIGLETGVIKNEHQVFKWDGKPRAMKQWERDLTLRGAIQVSAVPVFQQIAREVGEVRMQKYLKKFSYGNQNISGGIDKFWLEGQLRISAVNQVEFLESLYLNKLSASKENQLIVKEALVTEAAPEYLVHSKTGFSGVGTESNPGVAWWVGWVEKETEVYFFAFNMDIDNESKLPLRKSIPTKIMESEGII