6r5f A 3.25 BS01 JSW A 1 K45 M67 L70 V76 L78 M92 L129 H136 I154 A155 D156 L157 S161 F162 K22 M41 L44 V50 L52 M66 L103 H110 I128 A129 D130 L131 S135 F136 D138 K140 E142 N143 D156 T189 D112 K114 E116 N117 D130 T147 2.7.11.1 0004672,0005524,0006468 -logKd/Ki=7.70, IC50=20nM Q13546 31013427 301 VIKMKSSDSLAFHRTQGLMIMKTGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEETLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE