6pz1 A 2.65 BS01 HEM A 1 S167 V170 F214 I217 F226 A264 F270 R343 H346 I349 Y353 I354 G380 T382 F387 V391 S155 V158 F202 I205 F214 A252 F258 R331 H334 I337 Y341 I342 G355 T357 F362 V366 1.13.11.52 0002376,0002666,0002678,0002830,0004833,0005737,0005829,0006569,0006954,0007565,0009055,0016702,0019441,0019805,0020037,0030485,0032421,0032496,0032693,0032735,0033555,0033754,0034276,0034354,0036269,0042098,0042130,0043065,0046006,0046872,0051213,0070233,0070234 P14902 31682426 501 KEYHIDEEVGFALPNPQENLPDFYNDWMFIAKHLPDLIESGQLRERVEKLNMLSIDHLTDHKSQRLARLVLGCITMAYVWGKGHGDVRKVLPRNIAVPYCQLSKKLELPPILVYADCVLANWKKKDPNKPLTYENMDVLFSFRDGDCSKGFFLVSLLVEIAAASAIKVIPTVFKAMQMQERDTLLKALLEIASCLEKALQVFHQIHDHVNPKAFFSVLRIYLSGWKGNPQLSDGLVYEGFWEDPKEFAGGSAGQSSVFQCFDVLLGIQQTAGGGHAAQFLQDMRRYMPPAHRNFLCSLESNPSVREFVLSKGDAGLREAYDACVKALVSLRSYHLQIVTKYILIPASQQPAKGTGGTDLMNFLKTVRSTTEKSLLK 6pz1 A 2.65 BS02 AOJ A 1 Y126 F163 F226 G262 S263 A264 G378 T379 Y114 F151 F214 G250 S251 A252 G353 T354 1.13.11.52 0002376,0002666,0002678,0002830,0004833,0005737,0005829,0006569,0006954,0007565,0009055,0016702,0019441,0019805,0020037,0030485,0032421,0032496,0032693,0032735,0033555,0033754,0034276,0034354,0036269,0042098,0042130,0043065,0046006,0046872,0051213,0070233,0070234 IC50=410nM, Kd=14000nM P14902 31682426 502 KEYHIDEEVGFALPNPQENLPDFYNDWMFIAKHLPDLIESGQLRERVEKLNMLSIDHLTDHKSQRLARLVLGCITMAYVWGKGHGDVRKVLPRNIAVPYCQLSKKLELPPILVYADCVLANWKKKDPNKPLTYENMDVLFSFRDGDCSKGFFLVSLLVEIAAASAIKVIPTVFKAMQMQERDTLLKALLEIASCLEKALQVFHQIHDHVNPKAFFSVLRIYLSGWKGNPQLSDGLVYEGFWEDPKEFAGGSAGQSSVFQCFDVLLGIQQTAGGGHAAQFLQDMRRYMPPAHRNFLCSLESNPSVREFVLSKGDAGLREAYDACVKALVSLRSYHLQIVTKYILIPASQQPAKGTGGTDLMNFLKTVRSTTEKSLLK