6pno A 1.82 BS01 ORM A 1 C32 F34 Y229 C30 F32 Y227 1.20.4.2,1.8.5.1,2.5.1.18 0004364,0005515,0005737,0005829,0006749,0010880,0010881,0014810,0016491,0016740,0019852,0042178,0045174,0050610,0060315,0060316,0070062,0071243,0098869 -logKd/Ki=5.32, Ki=4.8uM Ki=4800nM, IC50=70nM P78417 32105470 1001 GESARSLGKGSAPPGPVPEGSIRIYSMRFCPFAERTRLVLKAKGIRHEVININLKNKPEWFFKKNPFGLVPVLENSQGQLIYESAITCEYLDEAYPGKKLLPDDPYEKACQKMILELFSKVPSLVGSFIRSQNKEDYAGLKEEFRKEFTKLEEVLTNKKTTFFGGNSISMIDYLIWPWFERLEAMKLNECVDHTPKLKLWMAAMKEDPTVSALLTSEKDWQGFLELYLQNSPEACDYGL