6oi8 A 2.5 BS01 MQV A 1 I157 K159 M169 E201 Y203 L204 H209 Q233 E276 L278 E288 I437 I157 K159 M164 E196 Y198 L199 H204 Q228 E271 L273 E283 I432 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D191 H204 R230 T269 E271 E283 N285 R287 E291 R333 6.3.4.14 0003824,0003989,0004075,0005524,0006633,0016874,0046872,2001295 -logKd/Ki=7.82, IC50<15nM P43873 31306011 502 MLEKVVIANRGEIALRILRACKELGIKTVAVHSTADRDLKHVLLADETICIGPAPSAKSYLNIPAIIAAAEVTGADAIHPGYGFLSENADFAEQVERSGFTFIGPTADVIRLMGDKVSAIKAMKKAGVPCVPGSDGPVSNDIAKNKEIAKRIGYPIIIKASGGMRVVRSEDALEESIAMTKAEAKAAFNNDMVYMEKYLENPRHVEIQVLADTHGNAVYLAERDCSMQRRHQKVVEEAPAPGITEEVRRDIGSRCANACVEIGYRGAGTFEFLYENGEFYFIEMNTRIQVEHPVTEMITGVDLVKEQLRIAAGLPISFKQEDIKVKGHAMECRINAEDPKTFLPSPGKVNHLHSPGGLGVRWDSHVYGGYTVPPHYDSMIAKLITYGDTREVAIRRMQNALSETIIDGIKTNIPLHELILEDENFQKGGTNIHYLEKKLG