6nzq A 2.11 BS01 LB4 A 1 L595 G598 V603 V640 K642 T687 E688 Y689 V690 E691 G693 R738 N739 L741 S758 L16 G19 V24 V35 K37 T82 E83 Y84 V85 E86 G88 R133 N134 L136 S153 N734 R738 N739 D759 N129 R133 N134 D154 2.7.10.2 0004672,0005524,0006468 ic50=0.3nM -logKd/Ki=9.52, IC50=0.3nM IC50=180nM P29597 31318208 4000 SFHRVDQKEITQLSHLGQGTRTNVYEGRLRELRVVLKVLDPSHHDIALAFYETASLMSQVSHTHLAFVHGVCVRGPENIMVTEYVEHGPLDVWLRRERGHVPMAWKMVVAQQLASALSYLENKNLVHGNVCGRNILLARLGLAEGTSPFIKLSDPGVGLGALSREERVERIPWLAPECLPSTAMDKWGFGATLLEICFDGEAPLQSRSPSEKEHFYQRQHRLPEPSCPQLATLTSQCLTYEPTQRPSFRTILRDLT