6nyh A 2.1 BS01 L8D A 1 I43 K45 M67 V75 V76 L78 L90 M92 H136 D156 L157 I26 K28 M50 V58 V59 L61 L73 M75 H119 D139 L140 D138 K140 E142 N143 D156 T189 D121 K123 E125 N126 D139 T160 2.7.11.1 0004672,0005524,0006468 Ki=21nM -logKd/Ki=7.68, Ki=21nM Q13546 31101885 301 NVIKMKSSDFLEKVSLAFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMAYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNEGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAIAEQQLIMAIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLE