6nvi A 2.117 BS01 XL7 A 1 V481 R483 A501 K503 E520 M524 I534 V550 C552 A553 G556 L610 A620 D621 V25 R27 A45 K47 E64 M68 I78 V94 C96 A97 G100 L152 A162 D163 D603 R607 N608 D621 D145 R149 N150 D163 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=8.59, IC50=2.6nM P22455 31413803 801 DLPLDPLWEFPRDRLVLGKPLGEQVVRAEAFGMDPARPDQASTVAVKMLKDNASDKDLADLVSEMEVMKLIGRHKNIINLLGVCTQEGPLYVIVECAAKGNLREFLRARRPPSEGPLSFPVLVSCAYQVARGMQYLESRKCIHRDLAARNVLVTEDNVMKIADFGLARGVLPVKWMAPEALFDRVYTHQSDVWSFGILLWEIFTLGGSPYPGIPVEELFSLLREGHRMDRPPHCPPELYGLMRECWHAAPSQRPTFKQLVEALDKVLLAV