6n79 A 2.27 BS01 KES A 1 L881 G882 G887 V889 A906 V938 M956 L959 E966 R1007 N1008 L1010 G1020 D1021 L16 G17 G22 V24 A41 V69 M83 L86 E93 R134 N135 L137 G147 D148 D1003 A1005 R1007 N1008 D1021 D130 A132 R134 N135 D148 2.7.10.2 0004672,0004713,0005524,0006468 Ki=0.21nM -logKd/Ki=9.68, Ki=0.21nM P23458 30981576 1201 DPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPNHIADLKKEIEILRNLYHENIVKYKGICTEGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIEKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK