6kzd A 1.708 BS01 DZ6 A 1 A570 K572 E588 L592 V601 F617 Y619 M620 L686 G696 D697 F698 A43 K45 E61 L65 V74 F90 Y92 M93 L147 G157 D158 F159 D679 R683 N684 D697 D140 R144 N145 D158 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 ic50=2.95nM -logKd/Ki=8.53, IC50=2.95nM Q16288 31271959 901 TYVQHIKRRDIVLKRELGEGAFGKVFLAECYNLSPTKDKMLVAVKALKDPTLAARKDFQREAELLTNLQHEHIVKFYGVCGDGDPLIMVFEYMKHGDLNKFLRAHGPDAGELGLSQMLHIASQIASGMVYLASQHFVHRDLATRNCLVGANLLVKIGDFGMSRDVYSTDYYRLHTMLPIRWMPPESIMYRKFTTESDVWSFGVILWEIFTYGKQPWFQLSNTEVIECITQGRVLERPRVCPKEVYDVMLGCWQREPQQRLNIKEIYKILHALGKATPIYLDI