6hkn A 2.33 BS01 G9E A 1 I61 Y66 A82 K84 I86 E102 L103 L106 L137 D138 M140 L189 D200 I8 Y10 A22 K24 I26 E42 L43 L46 L77 D78 M80 L129 D140 D182 K184 S186 N187 D200 T224 D122 K124 S126 N127 D140 T164 2.7.11.24 0004672,0004707,0005524,0006468 ic50=0.051uM -logKd/Ki=7.29, IC50=0.051uM IC50=51nM Q13164 30563338 1001 EYEIIETIAYGVVSSARRQQVAIKKIPNAFDVVTNAKRTLRELKILKHFKHDNIIAIKDILRPTVPYGEFKSVYVVLDLMESDLHQIIHSSQPLTLEHVRYFLYQLLRGLKYMHSAQVIHRDLKPSNLLVNENCELKIGDFGMARGLCTSPAEHQYFMTEYVATRWYRAPELMLSLHEYTQAIDLWSVGCIFGEMLARRQLFPGKNYVHQLQLIMMVLGTPSPAVIQAVGAERVRAYIQSLPPRQPVPWETVYPGADRQALSLLGRMLRFEPSARISAAAALRHPFLAKYHDPDDEPDCAPPFDFAFDREALTRERIKEAIVAEIEDFHARRE