6gvx A 2.24 BS01 TAK A 1 A38 L86 E87 C89 P90 G91 L139 A40 L85 E86 C88 P89 G90 L138 D132 K134 N137 D150 S171 D131 K133 N136 D149 S163 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 Ki=24nM -logKd/Ki=7.62, Ki=24nM Q14680 31108049 402 PLGSMKDYDELLKYYELHETIGTFAKVKLACHILTGEMVAIKIMDKNTDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCAKPKGNKCGSLAYAAPELIQGKGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR