6gk9 A 2.54 BS01 F2K A 1 G120 I132 V159 I179 K181 G121 I133 V154 I174 K176 1.1.1.205 0000166,0003824,0003938,0005524,0006164,0006177,0006183,0016491,0042802,0046872 IC50=4000nM Q9HXM5 30769241 501 HMLRISQEALTFDDVLLIPGYSEVLPKDVSLKTRLTRGIELNIPLVSAAMDTVTEARLAIAMAQEGGIGIIHKNMGIEQQAAEVRKVKKHETAIVRDPVTVTPSTKIIELLQMAREYGFSGFPVVEQGELVGIVTGRDLRDTVAAIMTPKDKLVTAREGTPLEEMKAKLYENRIEKMLVVDENFYLRGLVTFRDIEKAKTYPLASKDEQGRLRVGAAVGTGADTGERVAALVAAGVDVVVVDTAHGHSKGVIERVRWVKQTFPDVQVIGGNIATAEAAKALAEAGADAVKVGIGPGSCTTRIVAGVGVPQISAIANVAAALEGTGVPLIADGGIRFSGDLAKAMVAGAYCVMMGSMFAGTEEAPGEIELFQGRSYKSYRVPYKGALSAIVHQLMGGLRAAMGYTGSADIQQMRTQPQFVRITGA