6gcx A 1.553 BS01 EUW A 1 R426 L501 C502 T503 G505 L553 L567 R14 L87 C88 T89 G91 L139 L153 D546 A548 R550 N551 D564 D132 A134 R136 N137 D150 2.7.10.2 0004672,0004713,0005524,0006468 ic50=0.6nM -logKd/Ki=9.22, IC50=0.6nM Q00944 29897729 701 RDYEIQRERIELGRCIGEGQFGDVHQGIYMSPENPAMAVAIKTCKNSDSVREKFLQEALTMRQFDHPHIVKLIGVITENPVWIIMELCTLGELRSFLQVRKFSLDLASLILYAYQLSTALAYLESKRFVHRDIAARNVLVSATDCVKLGDFGLSRLPIKWMAPESINFRRFTSASDVWMFGVCMWEILMHGVKPFQGVKNNDVIGRIENGERLPMPPNCPPTLYSLMTKCWAYDPSRRPRFTELKAQLSTILEEEKLQ