6fyl A 1.95 BS01 3NG A 1 L169 G170 E171 F174 V177 A191 K193 F243 L246 L297 V326 D327 L26 G27 E28 F31 V34 A48 K50 F100 L103 L154 V183 D184 2.7.12.1 0004672,0005524,0006468 ic50=7nM -logKd/Ki=8.15, IC50=7nM IC50=4.0nM P49760 29985556 501 EDDAEGHLIYHVGDWLQERYEIVSTLGEGTFGRVVQCVDHRRGGARVALKIIKNVEKYKEAARLEINVLEKINEKDPDNKNLCVQMFDWFDYHGHMCISFELLGLSTFDFLKDNNYLPYPIHQVRHMAFQLCQAVKFLHDNKLTHTDLKPENILFVNSDYELTYNLEKKRDERSVKSTAVRVVDFGSATFDHEHHSTIVSTRHYRAPEVILELGWSQPCDVWSIGCIIFEYYVGFTLFQTHDNREHLAMMERILGPIPSRMIRKTRKQKYFYRGRLDWDENTSAGRYVRENCKPLRRYLTSEAEEHHQLFDLIESMLEYEPAKRLTLGEALQHPFFARLR