6cby A 2.55 BS01 ZN A 1 C52 C74 C78 C48 C70 C74 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 Q9NRG4 31415173 1001 GLGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLEFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEIES 6cby A 2.55 BS02 ZN A 2 C65 C68 H86 C90 C61 C64 H82 C86 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 Q9NRG4 31415173 1002 GLGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLEFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEIES 6cby A 2.55 BS03 ZN A 3 C209 C262 C264 C267 C205 C258 C260 C263 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 Q9NRG4 31415173 1003 GLGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLEFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEIES 6cby A 2.55 BS04 EW4 A 1 K17 H137 C181 N182 G183 F184 N206 H207 Y240 Y258 F260 E263 K13 H133 C177 N178 G179 F180 N202 H203 Y236 Y254 F256 E259 2.1.1.-,2.1.1.354 0000122,0000993,0002039,0005515,0005634,0005654,0005737,0005829,0006325,0006338,0007507,0008168,0008285,0016278,0016279,0018026,0018027,0032259,0042054,0043516,0046872,0046975,0140938,0140999,1901796 IC50=1300nM Q9NRG4 31415173 1004 GLGGLERFCSPGKGRGLRALQPFQVGDLLFSCPAYAYVLTVNERGNHCEYCFTRKEGLSKCGRCKQAFYCNVECQKEDWPMHKLECSPMVVFGENWNPSETVRLTARILAKQKIHPERTPSEKLLAVKEFESHLDKLDNEKKDLIQSDIAALHHFYSKHLEFPDNDSLVVLFAQVNCNGFTIEDEELSHLGSAIFPDVALMNHSCCPNVIVTYKGTLAEVRAVQEIKPGEEVFTSYIDLLYPTEDRNDRLRDSYFFTCECQECTTKDKDKAKVEIRKLSDPPKAEAIRDMVRYARNVIEEFRRAKHYKSPSELLEICELSQEKMSSVFEDSNVYMLHMMYQAMGVCLYMQDWEGALQYGQKIIKPYSKHYPLYSLNVASMWLKLGRLYMGLEHKAAGEKALKKAIAIMEVAHGKDHPYISEIKQEIES