5zz4 A 2.9 BS01 9M3 A 1 L408 G411 Q412 A428 K430 Y476 M477 N479 G480 D521 N526 L528 L542 S543 Y551 L14 G17 Q18 A34 K36 Y82 M83 N85 G86 D127 N132 L134 L148 S149 Y157 D521 R525 N526 D539 D127 R131 N132 D145 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=9.17, IC50=0.67nM IC50=0.670000nM Q06187 30216722 701 WEIDPKDLTFLKELGTGQFGVVKYGKWRGQYDVAIKMIKEGSMSEDEFIEEAKVMMNLSHEKLVQLYGVCTKQRPIFIITEYMANGCLLNYLREMRHRFQTQQLLEMCKDVCEAMEYLESKQFLHRDLAARNCLVNDQGVVKVSDFGLSRYVLDDEYTSSVGSKFPVRWSPPEVLMYSKFSSKSDIWAFGVLMWEIYSLGKMPYERFTNSETAEHIAQGLRLYRPHLASEKVYTIMYSCWHEKADERPTFKILLSNILDVM