5zt1 A 3.114 BS01 MG B 4 Y126 S127 Y46 S47 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 P0A1C1 30013545 507 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI 5zt1 A 3.114 BS02 AGS A 1 G162 G164 K165 T166 F167 F339 Y412 G82 G84 K85 T86 F87 F255 Y313 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 -logKd/Ki=4.67, Kd=21.23uM P0A1C1 30013545 502 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI 5zt1 A 3.114 BS03 MG A 1 E188 S250 R253 E108 S170 R173 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 P0A1C1 30013545 504 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI 5zt1 A 3.114 BS04 MG A 2 K141 V142 Q410 K61 V62 Q311 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 P0A1C1 30013545 505 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI 5zt1 A 3.114 BS05 MG A 3 G164 K165 G84 K85 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 P0A1C1 30013545 506 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI 5zt1 A 3.114 BS06 MG A 4 R320 L323 G325 R350 R236 L239 G241 R266 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 P0A1C1 30013545 507 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI 5zt1 A 3.114 BS07 MG A 5 T231 L285 Y302 T151 L205 Y222 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 P0A1C1 30013545 508 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI 5zt1 A 3.114 BS08 MG A 6 T252 D313 L315 T172 D229 L231 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 P0A1C1 30013545 509 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI 5zt1 A 3.114 BS09 MG A 7 E235 R238 E155 R158 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 P0A1C1 30013545 510 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI 5zt1 A 3.114 BS10 MG A 8 S297 T299 S217 T219 K165 E188 R189 R350 K85 E108 R109 R266 7.4.2.8 0005524,0005737,0009058,0016887,0030254,0030257 P0A1C1 30013545 511 SHMHTQVGRGLLGAVVNPLGEVTDKFAVTDNSEILYRPVDNAPPLYSERAAIEKPFLTGIKVIDSLLTCGEGQRMGIFASAGCGKTFLMNMLIEHSGADIYVIGLIGERGREVTETVDYLKNSEKKSRCVLVYATSDYSSVDRCNAAYIATAIAEFFRTEGHKVALFIDSLTRYARALRDVALAAGESPARRGYPVSVFDSLPRLLERPGKLKAGGSITAFYTVLLEADPLAEEVRSILDGHIYLSRNLAQKGQFPAIDSLKSISRVFTQVVDEKHRIMAAAFRELLSEIEELRTIKIYNKISVVESFLKQDYRLGFTYEQTMELIGETI