5yu9 A 1.95 BS01 1E8 A 1 L718 G719 A743 K745 M766 M790 M793 C797 R841 L844 T854 D855 F856 L19 G20 A44 K46 M63 M87 M90 C94 R138 L141 T151 D152 F153 D837 A839 R841 N842 D855 D134 A136 R138 N139 D152 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=6.74, Kd=0.18uM IC50=0.5nM, Kd=6.9nM P00533 27626175 1101 NQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLIMQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDERMHLPSPTDSNFYRALMDEEDMDDVVDADEYL