5x02 A 2.401 BS01 F6M A 1 L616 V624 A642 K644 V675 F691 E692 Y693 C694 C695 Y696 L818 C828 F830 L44 V52 A70 K72 V103 F119 E120 Y121 C122 C123 Y124 L176 C186 F188 D811 R815 N816 D829 D169 R173 N174 D187 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 -logKd/Ki=9.85, IC50=0.14nM P36888 29187377 1001 ESQLQMVQVTGSSDNEYFYVDFREYEYDLKWEFPRENLEFGKVLGSGAFGKVMNATAYGISKTGVSIQVAVKMLKEKADSSEREALMSELKMMTQLGSHENIVNLLGACTLSGPIYLIFEYCCYGDLLNYLRSKREKFSVLTFEDLLCFAYQVAKGMEFLEFKSCVHRDLAARNVLVTHGKVVKICDFGLARDIMSDSNYVVRGNARLPVKWMAPESLFEGIYTIKSDVWSYGILLWEIFSLGVNPYPGIPVDANFYKLIQNGFKMDQPFYATEEIYIIMQSCWAFDSRKRPSFPNLTSFLGCQL