5w8j A 1.55 BS01 9Y7 A 1 Q99 L108 N137 P138 D140 I141 R168 E191 H192 T247 L322 Q97 L106 N135 P136 D138 I139 R166 E189 H190 T245 L320 R105 D165 R168 H192 R103 D163 R166 H190 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 Kd=370nM -logKd/Ki=6.43, Kd=370nM IC50=>57000nM, EC50=3530nM, Kd=370nM P00338 29120638 501 ATLKDQLIYNLLKQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF 5w8j A 1.55 BS02 9Y7 A 2 V25 G26 D51 V52 K80 Y82 A95 G96 I115 F118 I119 V23 G24 D49 V50 K78 Y80 A93 G94 I113 F116 I117 R105 D165 R168 H192 R103 D163 R166 H190 1.1.1.27 0003824,0004459,0005515,0005634,0005737,0005739,0005829,0006089,0006090,0006096,0016020,0016491,0016616,0019752,0042802,0045296,0070062,1990204 Kd=370nM -logKd/Ki=6.43, Kd=370nM IC50=>57000nM, EC50=3530nM, Kd=370nM P00338 29120638 502 ATLKDQLIYNLLKQTPQNKITVVGVGAVGMACAISILMKDLADELALVDVIEDKLKGEMMDLQHGSLFLRTPKIVSGKDYNVTANSKLVIITAGARQQEGESRLNLVQRNVNIFKFIIPNVVKYSPNCKLLIVSNPVDILTYVAWKISGFPKNRVIGSGCNLDSARFRYLMGERLGVHPLSCHGWVLGEHGDSSVPVWSGMNVAGVSLKTLHPDLGTDKDKEQWKEVHKQVVESAYEVIKLKGYTSWAIGLSVADLAESIMKNLRRVHPVSTMIKGLYGIKDDVFLSVPCILGQNGISDLVKVTLTSEEEARLKKSADTLWGIQKELQF