5vcy A 1.56 BS01 DB8 A 1 L116 A137 V138 K139 V171 L185 T187 C190 G191 P192 F240 L50 A71 V72 K73 V105 L119 T121 C124 G125 P126 F174 D233 K235 N238 D251 D270 D167 K169 N172 D185 D204 2.7.11.1 0004672,0005524,0006468 Kd=270nM -logKd/Ki=6.57, Kd=270nM Ki=13nM, IC50=704nM, Kd=350nM Q99640 28792760 401 DLGTENLYFQLQPRRVSFRGEASETLQSPGYDPSRPESFFQQSFQRLSRLGHGSYGEVFKVRSKEDGRLYAVKRSMSPFRGPKDRARKLAEVGSHEKVGQHPCCVRLEQAWEEGGILYLQTELCGPSLQQHCEAWGASLPEAQVWGYLRDTLLALAHLHSQGLVHLDVKPANIFLGPRGRCKLGDFGLLVELGTAGAGEVQEGDPRYMAPELLQGSYGTAADVFSLGLTILEVACNMELPHGGEGWQQLRQGYLPPEFTAGLSSELRSVLVMMLEPDPKLRATAEALLALPVLRQP