5uit A 1.84 BS01 8CD A 1 M192 E194 G195 A211 Y262 Y264 M265 A315 N316 L318 S328 M31 E33 G34 A50 Y95 Y97 M98 A148 N149 L151 S161 D311 K313 A315 N316 D329 T351 D144 K146 A148 N149 D162 T179 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=4.6nM -logKd/Ki=8.34, IC50=4.6nM IC50=4.60nM Q9NWZ3 28498658 501 DTRFHSFSFYELKNVTNNFDERPISVGGNKMGEGGFGVVYKGYVNNTTVAVKKLTTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT