5uis A 2.5 BS01 8C1 A 1 E194 V200 A211 Y262 Y264 M265 A315 N316 L318 E30 V34 A45 Y85 Y87 M88 A138 N139 L141 D311 K313 A315 N316 D329 T351 D134 K136 A138 N139 D152 T166 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 ic50=146nM -logKd/Ki=6.84, IC50=146nM IC50=146nM Q9NWZ3 28498658 800 FHSFSFYELKNVTNNFDERPISVGGNKMGEGGVVYKGYVNNTTVAVKKLKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARAMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMT