5uiq A 2.64 BS01 8BV A 1 M192 V200 A211 Y262 M265 L318 M23 V31 A40 Y78 M81 L134 D311 K313 A315 N316 D329 T351 D127 K129 A131 N132 D145 T163 2.7.11.1 0000287,0004672,0004674,0005524,0006468,0007165 -logKd/Ki=4.26, IC50=55.056uM IC50=55000nM Q9NWZ3 28498658 501 RFHSFSFYELKNVTNNFDERPKMGEGGFGVVYKGYVTTVAVKKLAAKQQFDQEIKVMAKCQHENLVELLGFSSDCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGINFLHENHHIHRDIKSANILLDEAFTAKISDFGLARASQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDKKMNDADSTSVEAMYSVASQCLHEKKNKRPDIKKVQQLLQEMTA