5tt7 A 1.77 BS01 7KF A 1 A400 M448 E449 M450 G454 P455 R498 L501 S511 D512 A40 M83 E84 M85 G89 P90 R133 L136 S146 D147 D494 A496 R498 N499 D512 K533 D129 A131 R133 N134 D147 K168 2.7.10.2 0004672,0004713,0005524,0006468 ic50=13nM -logKd/Ki=7.89, IC50=13nM IC50=13nM, EC50=35nM P43405 27839918 901 IRPKEVYLDRKLLTLEDKELGSGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNHHHH