5tq5 A 2.3 BS01 7GX A 1 L855 A880 E898 M929 E930 Y931 L932 P933 G935 L983 D994 F995 L15 A40 E58 M89 E90 Y91 L92 P93 G95 L143 D154 F155 D976 A978 R980 N981 D994 S1016 D136 A138 R140 N141 D154 S176 2.7.10.2 0004672,0004713,0005524,0006468 ic50=58.8nM -logKd/Ki=7.23, IC50=58.8nM IC50=59nM O60674 27983835 4000 PTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQSIVTHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA