5teh A 2.99 BS01 S56 A 1 C281 A293 E310 M314 Y340 D404 C26 A38 E55 M59 Y85 D149 D386 R388 A390 N391 D404 F424 D131 R133 A135 N136 D149 F152 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=7.55, IC50=28nM P00523 600 AKDAWEIPRESLRLEVKLGQGCFGECWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL