5t68 A 2.93 BS01 77V A 1 L377 A400 M450 A451 L453 G454 L501 L15 A38 M83 A84 L86 G87 L134 D494 A496 R498 N499 D512 K533 D127 A129 R131 N132 D145 K162 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=7.64, IC50=0.023uM IC50=23nM, EC50=34nM P43405 27789138 701 VYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVNEG