5op5 A 1.9 BS01 3FE A 1 V23 A36 M84 E85 L86 A87 L137 D148 V20 A33 M73 E74 L75 A76 L126 D137 D130 K132 H134 N135 D148 T170 D119 K121 H123 N124 D137 T159 2.7.11.1 0000077,0004672,0004674,0005524,0006468 Ki=0.216uM -logKd/Ki=6.67, Ki=0.216uM O14757 29023112 301 PFVEDWDLVQTLGEGAYGEVQLAVNRVTEEAVAVKIVDMNIKKEICILKMLNHENVIKFYGHRREGNIQYLFMELASGGSLFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPHNLLLDERDNLKIADYSLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK